Potent and Selective KDM5 Inhibitor Stops Cellular Demethylation of H3K4me3 at Transcription Start Sites and Proliferation of MM1S Myeloma Cells

Tumber A., Nuzzi A., Hookway ES., Hatch SB., Velupillai S., Johansson C., Kawamura A., Savitsky P., Yapp C., Szykowska A., Wu N., Bountra C., Strain-Damerell C., Burgess-Brown NA., Ruda GF., Fedorov O., Munro S., England KS., Nowak RP., Schofield CJ., La Thangue NB., Pawlyn C., Davies F., Morgan G., Athanasou N., Müller S., Oppermann U., Brennan PE.

DOI

10.1016/j.chembiol.2017.02.006

Type

Journal article

Journal

Cell Chemical Biology

Publisher

Elsevier BV

Publication Date

03/2017

Volume

24

Pages

371 - 380

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