Design, Synthesis and Characterization of Covalent KDM5 Inhibitors

Vazquez-Rodriguez S., Wright M., Rogers CM., Cribbs AP., Velupillai S., Philpott M., Lee H., Dunford JE., Huber KVM., Robers MB., Vasta JD., Thezenas M-L., Bonham S., Kessler B., Bennett J., Fedorov O., Raynaud F., Donovan A., Blagg J., Bavetsias V., Oppermann U., Bountra C., Kawamura A., Brennan PE.

DOI

10.1002/anie.201810179

Type

Journal article

Journal

Angewandte Chemie International Edition

Publisher

Wiley

Publication Date

08/01/2019

Volume

58

Pages

515 - 519

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