Crystallographic fragment screening and deep mutational scanning of Zika virus NS2B-NS3 protease enable development of resistance-resilient inhibitors

Ni X., Richardson B., Godoy AS., Ferla M., Kikawa C., Scheen J., Hannon W., Capkin E., Lahav N., Balcomb B., Marples P., Fairhead M., Wang S., Williams E., Tomlinson CWE., Aschenbrenner JC., Lithgo R., Winokan M., Giroud C., Chandran A., Walsh M., Thompson W., Bloom J., Barr H., Kirkegaard K., Koekemoer L., Fearon D., Evans M., von Delft F.

DOI

10.1101/2024.04.29.591502

Type

Preprint

Publication Date

2024-01-01T00:00:00+00:00

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