Rational discovery of therapeutic PAK1 allosteric activators

He Y., Bae JSH., Nowak E., Outeiral C., Nissley DA., Tumber A., Berridge G., Salah E., Wang Y., He W., Zhang H., Chen T., Tusk S., Mathea S., Wang Y-J., Grassam-Rowe A., Kukura P., Schofield CJ., O’Brien DP., Pierangelini A., Churchill GC., Lanyon-Hogg T., Ke Y., Xu C., Ye T., Watkins H., Ying L., Koschinski A., Solaro RJ., Tan X., Bolla JR., Wang X., Knapp S., Deane CM., Zaccolo M., Nowotny M., Lei M.

DOI

10.1016/j.cell.2026.03.008

Type

Journal article

Publisher

Elsevier BV

Publication Date

2026-03-01T00:00:00+00:00

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