Elisabeth Mira Rothweiler
Postdoctoral Researcher
Recent publications
A BRET biosensor for measuring uncompetitive engagement of PRMT5 complexes in cells
Journal article
Rothweiler EM. et al, (2025), Nature Communications, 16
Phenomics‐Based Discovery of Novel Orthosteric Choline Kinase Inhibitors
Journal article
Bauer LG. et al, (2025), Angewandte Chemie International Edition, 64
A Live Cell BRET Probe to Quantify PRMT5-MTA Uncompetitive Target Engagement
Preprint
Rothweiler E. et al, (2025)
Covalent Inhibitors of KEAP1 with Exquisite Selectivity
Journal article
Fejes I. et al, (2024), Journal of Medicinal Chemistry, 67, 21208 - 21222
Abstract A005: A live cell PRMT5 NanoBRET™ target engagement assay querying competitive and uncompetitive modes of inhibition
Journal article
Teske KA. et al, (2024), Molecular Cancer Therapeutics, 23, A005 - A005
